| Family | Receptor | Species | Host Cell | Cell Line | Division Arrested Cells | Membranes |
|---|---|---|---|---|---|---|
| Zinc | GPR39 | Human | HEK293T | H1099 | DH1099 | MH1099 |
| Vasopressin/ Oxytocin | OT | Human | CHO-K1 | C1299-1 | DC1299-1 | MC1299-1 |
| Vasopressin/ Oxytocin | V1A | Human | CHO-K1 | C1042-1 | DC1042-1 | MC1042-1 |
| Vasopressin/ Oxytocin | V1B | Human | CHO-K1 | C1043-1 | DC1043-1 | MC1043-1 |
| Vasopressin/ Oxytocin | V2 | Human | CHO-K1 | C1044-1 | DC1044-1 | MC1044-1 |
| Vasopressin/ Oxytocin | V2 | dog | CHO-K1 | Cd1044-1 | DCd1044-1 | MCd1044-1 |
| Vasoactive Intestinal Peptide | PAC1 | Human | HEK293T | C1415 | DC1415 | MC1415 |
| Vasoactive Intestinal Peptide | VPAC1 | Human | CHO-K1 | C1292-1 | DC1292-1 | MC1292-1 |
| Vasoactive Intestinal Peptide | VPAC2 | Human | HEK293T | C1293 | DC1293 | MC1293 |
| Urotensin | UT | Rat | CHO dhfr- | C1035-1 | DC1035-1 | MC1035-1 |
| Urotensin | UT | Human | HEK293T | C1035-1a | DC1035-1a | DC1035-1a |
| Trace amine | TA1 | Rat | HEK293T | C1357 | DC1357 | MC1357 |
| Trace amine | TA1 | Human | HEK293T | C1357a | DC1357a | MC1357a |
| Thyrotropin-Releasing Hormone | TRH | Human | HEK293T | |||
| Tachykinin | NK1 | Human | HEK293T | C1303 | DC1303 | MC1303 |
| Tachykinin | NK2 | Human | HEK293T | C1304 | DC1304 | MC1304 |
| Tachykinin | NK3 | Human | HEK293T | C1305 | DC1305 | MC1305 |
| Somatostatin | sst1 | Human | CHO-K1 | C1345-1a | DC1345-1a | MC1345-1a |
| Somatostatin | sst1 | Human | CHO-K1 Gα16 | CG1345-1 | DCG1345-1 | MCG1345-1 |
| Somatostatin | sst2 | Human | CHO-K1 | C1346-1 | DC1346-1 | MC1346-1 |
| Somatostatin | sst2 | Human | CHO-K1 Gα16 | CG1346-1 | DCG1346-1 | MCG1346-1 |
| Somatostatin | sst3 | Human | CHO-K1 | C1347-1 | DC1347-1 | MC1347-1 |
| Somatostatin | sst3 | Human | CHO-K1 Gα16 | CG1347-1 | DCG1347-1 | MCG1347-1 |
| Somatostatin | sst4 | Human | CHO-K1 | C1348-1 | DC1348-1 | MC1348-1 |
| Somatostatin | sst4 | Human | CHO-K1 | C1348-1a | DC1348-1a | MC1348-1a |
| Somatostatin | sst4 | Human | CHO-K1 Gα16 | CG1348-1 | DCG1348-1 | MCG1348-1 |
| Somatostatin | sst5 | Human | CHO-K1 | C1349-1 | DC1349-1 | MC1349-1 |
| Somatostatin | sst5 | Human | CHO-K1 Gα16 | CG1349-1 | DCG1349-1 | MCG1349-1 |
| Serotonin | 5-HT1A | Human | HEK293T | C1319 | DC1319 | MC1319 |
| Serotonin | 5-HT1A | Human | HEK293T | C1319a | DC1319a | MC1319a |
| Serotonin | 5-HT1B | Human | HEK293T | C1320 | DC1320 | MC1320 |
| Serotonin | 5-HT1B | Human | HEK293T Gαqi5 | CG1320 | DCG1320 | MCG1320 |
| Serotonin | 5-HT2A | Human | CHO-K1 | C1324-1 | DC1324-1 | MC1324-1 |
| Serotonin | 5-HT2A | mouse | HEK293T | Cm1324 | DCm1324 | MCm1324 |
| Serotonin | 5-HT2A | dog | HEK293T | Cd1324 | DCd1324 | MCd1324 |
| Serotonin | 5-HT2B | Human | CHO-K1 | C1325-1 | DC1325-1 | MC1325-1 |
| Serotonin | 5-HT2B | Human | HEK293T | C1325 | DC1325 | MC1325 |
| Serotonin | 5-HT2B | mouse | HEK293T | Cm1325 | DCm1325 | MCm1325 |
| Serotonin | 5-HT2C | Human | CHO-K1 | C1326-1 | DC1326-1 | MC1326-1 |
| Serotonin | 5-HT4 | Human | CHO-K1 | C1330-1 | DC1330-1 | MC1330-1 |
| Serotonin | 5-HT4 | Human | HEK293T | C1330 | DC1330 | MC1330 |
| Serotonin | 5-HT6 | Human | CHO-K1 | C1331-1 | DC1331-1 | MC1331-1 |
| Serotonin | 5-HT7 | Human | HEK293T | C1334 | DC1334 | MC1334 |
| Relaxin | RXFP1 | Human | HEK293T | C1287 | DC1287 | MC1287 |
| Relaxin | RXFP1 | Human | HEK293T | C1287NTa | DC1287NTa | MC1287NTa |
| Relaxin | RXFP1 | Human | HEK293T | C1287NTb | DC1287NTb | MC1287NTb |
| Relaxin | RXFP2 | Human | HEK293T | C1289NTa | DC1289NTa | MC1289NTa |
| Relaxin | RXFP2 | Human | HEK293T | C1289NTb | DC1289NTb | MC1289NTb |
| Relaxin | RXFP3 | Human | HEK293T | C1306 | DC1306 | MC1306 |
| Purinergic | GPR17 | Human | 1321N1 | C1076-3 | DC1076-3 | MC1076-3 |
| Purinergic | GPR17 | Human | 1321N1 | C1076-3a | DC1076-3a | MC1076-3a |
| Purinergic | P2Y1 | Human | 1321N1 | C1160-3 | DC1160-3 | MC1160-3 |
| Purinergic | P2Y2 | Human | 1321N1 | C1161-3 | DC1161-3 | MC1161-3 |
| Purinergic | P2Y2 | Rat | 1321N1 | Cr1161-3 | DCr1161-3 | MCr1161-3 |
| Purinergic | P2Y4 | Human | 1321N1 | C1162-3 | DC1162-3 | MC1162-3 |
| Purinergic | P2Y6 | Human | 1321N1 | C1164-3 | DC1164-3 | MC1164-3 |
| Purinergic | P2Y11 | Human | 1321N1 | C1169-3 | DC1169-3 | MC1169-3 |
| Purinergic | P2Y12 | Human | 1321N1 | C1170-3 | DC1170-3 | MC1170-3 |
| Purinergic | P2Y12 | Rat | CHO dhfr- | C1170-1 | DC1170-1 | MC1170-1 |
| Purinergic | P2Y13 | Human | 1321N1 | C1139-3 | DC1139-3 | MC1139-3 |
| Purinergic | P2Y14 | Human | HEK293T | C1057 | DC1057 | MC1057 |
| Purinergic | P2Y14 | Human | HEK293T Gαqi5 | CG1057 | DCG1057 | MCG1057 |
| Purinergic | P2Y14 | Rat | HEK293T Gαqi5 | CGr1057 | DCGr1057 | MCGr1057 |
| Purinergic | P2Y14 | monkey | HEK293T Gαqi5 | CGp1057 | DCGp1057 | MCGp1057 |
| Protease-Activated | PAR1 | Human | CHO-K1 | C1207-1 | DC1207-1 | MC1207-1 |
| Protease-Activated | PAR1 | Human | HeLa | C1207-7 | DC1207-7 | MC1207-7 |
| Protease-Activated | PAR2 | Human | HeLa | C1208-7 | DC1208-7 | MC1208-7 |
| Protease-Activated | PAR4 | Human | HeLa | C1210-7 | DC1210-7 | MC1210-7 |
| Prostanoid | DP1 | Human | HEK293T | C1200 | DC1200 | MC1200 |
| Prostanoid | DP2 | Human | HEK293T | H1105 | DH1105 | MH1105 |
| Prostanoid | DP2 | Human | HEK293T | H1105a | DH1105a | MH1105a |
| Prostanoid | EP1 | Human | HEK293T | C1201a | DC1201a | MC1201a |
| Prostanoid | EP2 | Human | HEK293T | C1202 | DC1202 | MC1202 |
| Prostanoid | EP3 | Human | CHO-K1 | C1203-1 | DC1203-1 | MC1203-1 |
| Prostanoid | EP3 | Human | CHO-K1 | C1203-1a | DC1203-1a | MC1203-1a |
| Prostanoid | EP3 | Human | CHO-K1 | C1203-1b | DC1203-1b | MC1203-1b |
| Prostanoid | EP3 | Human | CHO-K1 | C1203-1c | DC1203-1c | MC1203-1c |
| Prostanoid | EP3 | Human | CHO-K1 | C1203-1d | DC1203-1d | MC1203-1d |
| Prostanoid | EP4 | Human | HEK293T | C1204 | DC1204 | MC1204 |
| Prostanoid | FP | Human | HEK293T | C1205 | DC1205 | MC1205 |
| Prostanoid | IP1 | Human | CHO-K1 | C1206-1 | DC1206-1 | MC1206-1 |
| Prostanoid | TP | Human | HEK293T | C1365 | DC1365 | MC1365 |
| Prostanoid | TP | Human | HEK293T | H1365 | DH1365 | MH1365 |
| Prolactin-Releasing Peptide | PrRP | Human | CHO dhfr- | C1037 | DC1037 | MC1037 |
| Prokineticin | PK1 | Human | CHO-K1 | C1128-1 | DC1128-1 | MC1128-1 |
| Prokineticin | PK2 | Human | CHO-K1 | C1127-1a | DC1127-1a | MC1127-1a |
| Prokineticin | PK2 mutant | Human | CHO-K1 | C1127CT-1 | DC1127DCT-1 | MC1127MCT-1 |
| Platelet-Activating Factor | PAF | Human | HEK293T | C1218 | DC1218 | MC1218 |
| Parathyroid Hormone | PTH1 | Human | HEK293T | C1301 | DC1301 | MC1301 |
| Parathyroid Hormone | PTH2 | Human | HEK293T | H1302 | DH1302 | MH1302 |
| Oxysterol | EBI2 | Human | CHO-K1 Gαqi5 | CG1242-1 | DCG1242-1 | MCG1242-1 |
| Oxysterol | EBI2 | mouse | CHO-K1 Gαqi5 | CGm1242-1 | DCGm1242-1 | MCGm1242-1 |
| Oxysterol | EBI2 | mouse | CHO-K1 | Cm1242-1 | DCm1242-1 | MCm1242-1 |
| Orphan | GPR3 | Human | HEK293T | C1091 | DC1091 | MC1091 |
| Orphan | GPR35 | dog | HEK293TGα16 | CGd1096 | DCGd1096 | MCGd1096 |
| Orphan | GPR35 | Human | HEK293TGα16 | CG1096 | DCG1096 | MCG1096 |
| Orphan | GPR50 | Human | HEK293T | C1110 | DC1110 | MC1110 |
| Orphan | GPR142 | Human | HEK293T | C1286 | DC1286 | MC1286 |
| Orphan | MRGX1 | Human | CHO dhfr-Gαqi5 | C1256 | DC1256 | MC1256 |
| Orphan | MRGX2 | Human | HEK293T Gαqi5 | C1257 | DC1257 | MC1257 |
| Orexin | OX1 | Human | CHO-K1 | C1033-1 | DC1033-1 | MC1033-1 |
| Orexin | OX2 | Human | CHO-K1 | C1034-1 | DC1034-1 | MC1034-1 |
| Opioid | delta | Human | CHO-K1 | C1351-1 | DC1351-1 | MC1351-1 |
| Opioid | delta | Human | CHO-K1 Gαqi5 | CG1351-1 | DCG1351-1 | MCG1351-1 |
| Opioid | delta | Rat | CHO dhfr- | C1351 | DC1351 | MC1351 |
| Opioid | kappa | Human | CHO-K1 | C1352-1a | DC1352-1a | MC1352-1a |
| Opioid | kappa | Human | CHO-K1 Gαqi5 | CG1351-1 | DCG1351-1 | MCG1351-1 |
| Opioid | kappa | Human | HEK293T | C1352 | DC1352 | MC1352 |
| Opioid | kappa | Rat | CHO dhfr- | C1352-1 | DC1352-1 | MC1352-1 |
| Opioid | mu | Human | CHO-K1 | C1350-1a | DC1350-1a | MC1350-1a |
| Opioid | mu | Human | CHO-K1 Gαqi5 | CG1350-1 | DCG1350-1 | MCG1350-1 |
| Opioid | mu | Rat | CHO dhfr- | Cr1350-1 | DCr1350-1 | MCr1350-1 |
| Opioid | NOP | Human | CHO-K1 | C1354-1 | DC1354-1 | MC1354-1 |
| Opioid | NOP | Human | CHO-K1 Gαqi5 | CG1354-1 | DCG1354-1 | MCG1354-1 |
| Opioid | NOP | Human | HEK293T | C1354a | DC1354a | MC1354a |
| Opioid | NOP | Rat | CHO dhfr- | C1354 | DC1354 | MC1354 |
| Nicotinic Acid | GPR109A | Human | CHO-K1 | C1370-1 | DC1370-1 | MC1370-1 |
| Nicotinic Acid | GPR109B | Human | CHO-K1 | C1059-1 | DC1059-1 | MC1059-1 |
| Neurotensin | NTS1 | Human | CHO-K1 | C1276-1 | DC1276-1 | MC1276-1 |
| Neurotensin | NTS2 | Human | CHO-K1 | C1277-1 | DC1277-1 | MC1277-1 |
| Neurotensin | NTS2 | Human | HEK293T | C1277 | DC1277 | MC1277 |
| Neurotensin | NTS2 | Human | HEK293T | C1277a | DC1277a | MC1277a |
| Neuropeptide Y | Y1 | Human | CHO-K1 Gαqi5 | CG1273-1 | DCG1273-1 | MCG1273-1 |
| Neuropeptide Y | Y2 | Human | CHO-K1 Gαqi5 | CG1274-1 | DCG1274-1 | MCG1274-1 |
| Neuropeptide Y | Y2 | Rat | CHO-K1 | Cr1274-1 | DCr1274-1 | MCr1274-1 |
| Neuropeptide Y | Y4 | Human | CHO-K1 | C1300-1 | DC1300-1 | MC1300-1 |
| Neuropeptide Y | Y4 | Human | CHO-K1 Gαqi5 | CG1300-1 | DCG1300-1 | MCG1300-1 |
| Neuropeptide Y | Y5 | Human | HEK293T | C1275a | DC1275a | MC1275a |
| Neuropeptide Y | Y5 | Human | HEK293T Gαqi5 | CG1275 | DCG1275 | MCG1275 |
| Neuropeptide W/B | NPBW1 | Rat | HEK293T Gαqi5 | C1124-1 | DC1124-1 | MC1124-1 |
| Neuropeptide W/B | NPBW1 | Human | HEK293T Gαqi5 | C1124 | DC1124 | MC1124 |
| Neuropeptide W/B | NPBW2 | Human | HEK293T Gαqi5 | C1133 | DC1133 | MC1133 |
| Neuropeptide S | NPS | mouse | HEK293T | C1355-1 | DC1355-1 | MC1355-1 |
| Neuropeptide S | NPS | Human | HEK293T | C1355a | DC1355a | MC1355a |
| Neuropeptide S | NPS(2) | Human | HEK293T | C1356 | DC1356 | MC1356 |
| Neuropeptide S | NPSIle107 | Human | HEK293T | C1355-2 | DC1355-2 | MC1355-2 |
| Neuropeptide FF/AF | NPFF1 | Human | HEK293T | C1363 | DC1363 | MC1363 |
| Neuropeptide FF/AF | NPFF2 | Human | HEK293T | CG1364 | DCG1364 | MCG1364 |
| Neuromedin U | NMU1 | Human | HEK293T | C1122 | DC1122 | MC1122 |
| Neuromedin U | NMU2 | Human | HEK293T | C1213 | DC1213 | MC1213 |
| N-formylpeptide | FPR1 | Human | HEK293T Gαqi5 | CG1243 | DCG1243 | MCG1243 |
| Muscarinic | M1 | Human | CHO-K1 | C1022-1 | DC1022-1 | MC1022-1 |
| Muscarinic | M1 | Human | CHO-K1 | C1022-1a | DC1022-1a | MC1022-1a |
| Muscarinic | M2 | Human | CHO-K1 | C1023-1 | DC1023-1 | MC1023-1 |
| Muscarinic | M3 | Human | CHO-K1 | C1024-1 | DC1024-1 | MC1024-1 |
| Muscarinic | M3 | mouse | CHO-K1 | Cm1024-1 | DCm1024-1 | MCm1024-1 |
| Muscarinic | M3 | Rat | CHO-K1 | |||
| Muscarinic | M4 | Human | CHO-K1 | C1025-1 | DC1025-1 | MC1025-1 |
| Muscarinic | M4 | Human | CHO-K1 Gαqi5 | CG1025-1 | DCG1025-1 | MCG1025-1 |
| Muscarinic | M5 | Human | CHO-K1 | C1026-1 | DC1026-1 | MC1026-1 |
| Motilin | motilin | Human | HEK293T | H1297 | DH1297 | MH1297 |
| Metabotropic Glutamate | mGlu1 | Human | CHO-K1 | C1188-1 | DC1188-1 | MC1188-1 |
| Metabotropic Glutamate | mGlu2 | Human | HEK293T | C1189a | DC1189a | MC1189a |
| Metabotropic Glutamate | mGlu2 | Human | HEK293T Gαqi5 | HG1189 | DHG1189 | MHG1189 |
| Metabotropic Glutamate | mGlu2 | Rat | HEK293T Gαqi5 | HGr1189 | DHGr1189 | MHGr1189 |
| Metabotropic Glutamate | mGlu3 | Human | HEK293T Gαqi5 | CG1190 | DCG1190 | MCG1190 |
| Metabotropic Glutamate | mGlu4 | dog | CHO-K1 Gαqi5 | CGd1191-1 | DCGd1191-1 | MCGd1191-1 |
| Metabotropic Glutamate | mGlu4 | dog | HEK293T Gαqi5 | CGd1191 | DCGd1191 | MCGd1191 |
| Metabotropic Glutamate | mGlu4 | dog | HEK293T Gαqi5 | HGd1191 | DHGd1191 | MHGd1191 |
| Metabotropic Glutamate | mGlu4 | Human | HEK293T | C1191a | DC1191a | MC1191a |
| Metabotropic Glutamate | mGlu4 | Human | HEK293T Gαqi5 | CG1191 | DCG1191 | MCG1191 |
| Metabotropic Glutamate | mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1a | DHGm1191-1a | MHGm1191-1a |
| Metabotropic Glutamate | mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1b | DHGm1191-1b | MHGm1191-1b |
| Metabotropic Glutamate | mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1c | DHGm1191-1c | MHGm1191-1c |
| Metabotropic Glutamate | mGlu4 | mouse | CHO-K1 Gαqi5 | HGm1191-1d | DHGm1191-1d | MHGm1191-1d |
| Metabotropic Glutamate | mGlu4 | Rat | HEK293T | Cr1191 | DCr1191 | MCr1191 |
| Metabotropic Glutamate | mGlu5 | Human | HEK293T | C1192 | DC1192 | MC1192 |
| Metabotropic Glutamate | mGlu6 | Human | HEK293T | C1193 | DC1193 | MC1193 |
| Metabotropic Glutamate | mGlu6 | Human | HEK293T | CG1193 | DCG1193 | MCG1193 |
| Metabotropic Glutamate | mGlu7 | Human | HEK293T | C1194 | DC1194 | MC1194 |
| Metabotropic Glutamate | mGlu7 | Human | HEK293T | CG1194 | DCG1194 | MCG1194 |
| Metabotropic Glutamate | mGlu8 | Human | HEK293T | C1195 | DC1195 | MC1195 |
| Metabotropic Glutamate | mGlu8 | Human | HEK293T | C1195a | DC1195a | MC1195a |
| Metabotropic Glutamate | mGlu8 | Human | HEK293T | CG1195 | DCG1195 | MCG1195 |
| Metabotropic Glutamate | mGlu8 | Human | CHO-K1 | C1195-1a | DC1195-1a | MC1195-1a |
| Melatonin | MT1 | Human | CHO-K1 | C1223-1 | DC1223-1 | MC1223-1 |
| Melatonin | MT2 | Human | HEK293T Gαqi5 | C1224 | DC1224 | MC1224 |
| Melatonin | MT2 | mouse | HEK293T | Cm1224 | DCm1224 | MCm1224 |
| Melatonin | MT2 | Rat | HEK293T | Cr1224 | DCr1224 | MCr1224 |
| Melanocortin | MC1 | Human | HEK293T | C1340 | DC1340 | MC1340 |
| Melanocortin | MC4 | Human | HEK293T | H1343 | DH1343 | MH1343 |
| Melanin-ConcentRating Hormone | MCH1 | Human | HEK293T Gαqi5 | C1031-3 | DC1031-3 | MC1031-3 |
| Melanin-ConcentRating Hormone | MCH1 | Rat | HEK293T Gαqi5 | C1031-4 | DC1031-4 | MC1031-4 |
| Melanin-ConcentRating Hormone | MCH2 | Human | CHO dhfr- | C1032 | DC1032 | MC1032 |
| Lysophospholipid | LPA1 | Human | RH7777 | C1048-6 | DC1048-6 | MC1048-6 |
| Lysophospholipid | LPA1 | mouse | RH7777 | Cm1048-6A | DCm1048-6A | MCm1048-6A |
| Lysophospholipid | LPA1 | mouse | RH7777 | Cm1048-6B | DCm1048-6B | MCm1048-6B |
| Lysophospholipid | LPA1 | Rat | RH7777 | Cr1048-6A | DCr1048-6A | MCr1048-6A |
| Lysophospholipid | LPA1 | Rat | RH7777 | Cr1048-6B | DCr1048-6B | MCr1048-6B |
| Lysophospholipid | LPA2 | Human | RH7777 | C1050-6 | DC1050-6 | MC1050-6 |
| Lysophospholipid | LPA2 | Human | CHO-K1 | C1050-1 | DC1050-1 | MC1050-1 |
| Lysophospholipid | LPA3 | Human | RH7777 | C1053-6 | DC1053-6 | MC1053-6 |
| Lysophospholipid | LPA3 | Human | RH7777 | C1053-6a | DC1053-6a | MC1053-6a |
| Lysophospholipid | LPA4 | Human | CHO-K1 | C1087-1a | DC1087-1a | MC1087-1a |
| Lysophospholipid | LPA5 | Human | RH7777 | C1145-6 | DC1145-6 | MC1145-6 |
| Lysophospholipid | LPA5 | mouse | RH7777 | Cm1145-6 | DCm1145-6 | MCm1145-6 |
| Lysophospholipid | S1P1 | Human | CHO-K1 | C1047-1 | DC1047-1 | MC1047-1 |
| Lysophospholipid | S1P1 | Human | CHO-K1 Gαqi5 | CG1047-1 | DCG1047-1 | MCG1047-1 |
| Lysophospholipid | S1P2 | Human | CHO-K1 | C1051-1 | DC1051-1 | MC1051-1 |
| Lysophospholipid | S1P2 | Human | CHO-K1 Gαqi5 | CG1051-1 | DCG1051-1 | MCG1051-1 |
| Lysophospholipid | S1P3 | Human | RH7777 | C1049-6 | DC1049-6 | MC1049-6 |
| Lysophospholipid | S1P3 | Human | CHO-K1 | C1049-1 | DC1049-1 | MC1049-1 |
| Lysophospholipid | S1P3 | Human | CHO-K1 Gαqi5 | CG1049-1 | DCG1049-1 | MCG1049-1 |
| Lysophospholipid | S1P4 | Human | CHO-K1 Gαqi5 | CG1052-1 | DCG1052-1 | MCG1052-1 |
| Lysophospholipid | S1P5 | Human | CHO-K1 | C1054-1 | DC1054-1 | MC1054-1 |
| Lysophospholipid | S1P5 | Human | CHO-K1 Gαqi5 | CG1054-1 | DCG1054-1 | MCG1054-1 |
| Leukotriene/Lipoxin | ALX | Human | HEK293T | C1244 | DC1244 | MC1244 |
| Leukotriene/Lipoxin | BLT1 | Human | HEK293T | H1165a | DH1165a | MH1165a |
| Leukotriene/Lipoxin | BLT2 | Human | HEK293T | C1272 | DC1272 | MC1272 |
| Leukotriene/Lipoxin | BLT2 | Human | HEK293T | C1272A | DC1272A | MC1272A |
| Leukotriene/Lipoxin | BLT2 | monkey | HEK293T | Cp1272a | DCp1272a | MCp1272a |
| Leukotriene/Lipoxin | BLT2 | monkey | HEK293T | Cp1272 | DCp1272 | MCp1272 |
| Leukotriene/Lipoxin | BLT2 | mouse | HEK293T | Cm1272a | DCm1272a | MCm1272a |
| Leukotriene/Lipoxin | BLT2 | mouse | HEK293T | Cm1272 | DCm1272 | MCm1272 |
| Leukotriene/Lipoxin | CysLT1 | Human | HEK293T | C1308 | DC1308 | MC1308 |
| Leukotriene/Lipoxin | CysLT2 | Human | HEK293T | C1307 | DC1307 | MC1307 |
| Leukotriene/Lipoxin | OXE | Human | HEK293T | |||
| KiSS1-Derived Peptide | KiSS1 | Human | CHO dhfr- | C1036 | DC1036 | MC1036 |
| KiSS1-Derived Peptide | KiSS1 | Rat | CHO dhfr- | C1036-1 | DC1036-1 | MC1036-1 |
| Hydroxycarboxylic acid | GPR81 | Human | HEK293T | |||
| Histamine | H1 | Human | HEK293T | C1027 | DC1027 | MC1027 |
| Histamine | H1 | mouse | HEK293T | Cm1027 | DCm1027 | MCm1027 |
| Histamine | H2 | Human | HEK293T | C1028 | DC1028 | MC1028 |
| Histamine | H3 | Human | HEK293T | C1029 | DC1029 | MC1029 |
| Histamine | H3 | Human | HEK293T Gαqi5 | CG1029 | DCG1029 | MCG1029 |
| Histamine | H3 | mouse | HEK293T | Cm1029 | DCm1029 | MCm1029 |
| Histamine | H3 | mouse | CHO-K1 | Cm1029-1 | DCm1029-1 | MCm1029-1 |
| Histamine | H4 | Human | HEK293T | C1030 | DC1030 | MC1030 |
| Histamine | H4 | Human | HEK293T Gαqi5 | CG1030 | DCG1030 | MCG1030 |
| Histamine | H4 | mouse | HEK293T | Cm1030 | DCm1030 | MCm1030 |
| Histamine | H4 | mouse | HEK293T Gαqi5 | CGm1030 | DCGm1030 | MCGm1030 |
| Gonadotrophin-Releasing Hormone | GnRH | Human | HEK293T | C1283 | DC1283 | MC1283 |
| Glycoprotein Hormone | TSH | Human | HEK293T | H1177 | DH1177 | MH1177 |
| Glycoprotein Hormone | TSH | Rat | HEK293T | C1177-1 | DC1177-1 | MC1177-1 |
| Glucagon | GHRH | Human | HEK293T | C1291 | DC1291 | MC1291 |
| Glucagon | GIP | Human | HEK293T | C1290 | DC1290 | MC1290 |
| Glucagon | GLP-1 | Human | HEK293T | C1267 | DC1267 | MC1267 |
| Glucagon | GLP-2 | Human | HEK293T | C1268 | DC1268 | MC1268 |
| Glucagon | GLP-2 | Rat | HEK293T | Cr1268 | DCr1268 | MCr1268 |
| Glucagon | Glucagon | Human | HEK293T | C1266 | DC1266 | MC1266 |
| Glucagon | Glucagon | Human | HEK293T | C1266A | DC1266A | MC1266A |
| Glucagon | Secretin | Human | CHO-K1 | C1228-1 | DC1228-1 | MC1228-1 |
| Ghrelin | Ghrelin | Human | HEK293T | C1197b | DC1197b | MC1197b |
| Ghrelin | Ghrelin | Human | CHO-K1 | C1197-1 | DC1197-1 | MC1197-1 |
| Ghrelin | Ghrelin | mouse | HEK293T | Cm1197 | DCm1197 | MCm1197 |
| Galanin | GAL1 | Human | CHO-K1 Gαqi5 | CG1178-1 | DCG1178-1 | MCG1178-1 |
| Galanin | GAL1 | Human | HEK293T | C1178 | DC1178 | MC1178 |
| Galanin | GAL2 | Human | CHO-K1 | C1179-1 | DC1179-1 | MC1179-1 |
| Frizzled | SMO | Human | HEK293T | C1442 | DC1442 | MC1442 |
| Free Fatty Acid | GPR119 | Human | CHO-K1 | C1298-1a | DC1298-1a | MC1298-1a |
| Free Fatty Acid | GPR119 | Human | HEK293T | C1298 | DC1298 | MC1298 |
| Free Fatty Acid | GPR119 | mouse | CHO-K1 | Cm1298-1 | DCm1298-1 | MCm1298-1 |
| Free Fatty Acid | GPR120 | Human | HEK293T | C1294 | DC1294 | MC1294 |
| Free Fatty Acid | GPR120 | Human | HEK293T Gαqi5 | CG1294 | DCG1294 | MCG1294 |
| Free Fatty Acid | GPR120 | Human | CHO-K1 | C1294-1 | DC1294-1 | MC1294-1 |
| Free Fatty Acid | GPR120 | mouse | HEK293T Gαqi5 | CGm1294 | DCGm1294 | MCGm1294 |
| Free Fatty Acid | GPR120 | Rat | HEK293T | Cr1294 | DCr1294 | MCr1294 |
| Free Fatty Acid | GPR40 | cynomolgus monkey | CHO-K1 | Cpc1101-1 | DCpc1101-1 | MCpc1101-1 |
| Free Fatty Acid | GPR40 | dog | CHO-K1 | Cd1101-1 | DCd1101-1 | MCd1101-1 |
| Free Fatty Acid | GPR40 | Human | HEK293T | C1101 | DC1101 | MC1101 |
| Free Fatty Acid | GPR40 | Human | CHO-K1 | C1101-1 | DC1101-1 | MC1101-1 |
| Free Fatty Acid | GPR40 | Human | CHO-K1 | C1101-1A | DC1101-1A | MC1101-1A |
| Free Fatty Acid | GPR40 | mouse | HEK293T | Cm1101 | DCm1101 | MCm1101 |
| Free Fatty Acid | GPR40 | mouse | MIN6 | |||
| Free Fatty Acid | GPR40 | Rat | HEK293T | Cr1101 | DCr1101 | MCr1101 |
| Free Fatty Acid | GPR40 | Rat | CHO-K1 | Cr1101-1 | DCr1101-1 | MCr1101-1 |
| Free Fatty Acid | GPR40 | rhesus monkey | CHO-K1 | Cpr1101-1 | DCpr1101-1 | MCpr1101-1 |
| Free Fatty Acid | GPR41 | Human | HEK293T | C1102 | DC1102 | MC1102 |
| Free Fatty Acid | GPR41 | Human | CHO-K1 Gα16 | C1102-1 | DC1102-1 | MC1102-1 |
| Free Fatty Acid | GPR41 | Human | HEK293T Gαqi5 | CG1102 | DCG1102 | MCG1102 |
| Free Fatty Acid | GPR41 | mouse | CHO-K1 Gα16 | CGm1102-1 | DCGm1102-1 | MCGm1102-1 |
| Free Fatty Acid | GPR41 | Rat | HEK293T | Cr1102 | DCr1102 | MCr1102 |
| Free Fatty Acid | GPR43 | Human | HEK293T | C1104 | DC1104 | MC1104 |
| Free Fatty Acid | GPR43 | Human | CHO-K1 | C1104-1 | DC1104-1 | MC1104-1 |
| Free Fatty Acid | GPR43 | Human | CHO-K1 Gα16 | HG1104-1 | DHG1104-1 | MHG1104-1 |
| Free Fatty Acid | GPR43 | mouse | HEK293T | Cm1104 | DCm1104 | MCm1104 |
| Free Fatty Acid | GPR43 | Rat | HEK293T | Cr1104 | DCr1104 | MCr1104 |
| Free Fatty Acid | GPR43 | dog | CHO-K1 | Cd1104-1 | DCd1104-1 | MCd1104-1 |
| Free Fatty Acid | GPR43 | cynomolgus monkey | CHO-K1 | Cpc1101-1 | DCpc1101-1 | MCpc1101-1 |
| Free Fatty Acid | GPR43 | rhesus monkey | CHO-K1 | Cpr1101-1 | DCpr1101-1 | MCpr1101-1 |
| Free Fatty Acid | GPR84 | Human | CHO-K1 | C1137-1 | DC1137-1 | MC1137-1 |
| Free Fatty Acid | GPR84 | Human | CHO-K1 Gαqi5 | CG1137-1 | DCG1137-1 | MCG1137-1 |
| Endothelin | ETA | Human | CHO-K1 | C1216-1 | DC1216-1 | MC1216-1 |
| Endothelin | ETA | Rat | CHO-K1 | Cr1216-1 | DCr1216-1 | MCr1216-1 |
| Endothelin | ETB | Human | CHO-K1 | C1217-1 | DC1217-1 | MC1217-1 |
| Dopamine | D1 | Human | HEK293T | H1335 | DH1335 | MH1335 |
| Dopamine | D2 | Human | HEK293T | C1336 | DC1336 | MC1336 |
| Dopamine | D2 | Human | HEK293T | C1336a | DC1336a | MC1336a |
| Dopamine | D4 | Human | HEK293T | C1338 | DC1338 | MC1338 |
| Dopamine | D4 | Human | HEK293T Gαqi5 | CG1338 | DCG1338 | MCG1338 |
| Dopamine | D5 | Human | HEK293T | C1339 | DC1339 | MC1339 |
| Corticotrophin-Releasing Factor | CRF1 | Human | HEK293T | C1040 | DC1040 | MC1040 |
| Corticotrophin-Releasing Factor | CRF1 | Human | HEK293T Gαqi5 | CG1040 | DCG1040 | MCG1040 |
| Corticotrophin-Releasing Factor | CRF2 | Human | HEK293T | C1041 | DC1041 | MC1041 |
| Corticotrophin-Releasing Factor | CRF2 | Human | HEK293TGα16 | CG1041 | DCG1041 | MCG1041 |
| Citric Acid Cycle Intermediates | GPR91 | Human | CHO-K1 | C1144-1 | DC1144-1 | MC1144-1 |
| Citric Acid Cycle Intermediates | GPR99 | Human | CHO-K1 | C1132-1 | DC1132-1 | MC1132-1 |
| Cholecystokinin | CCK1 | Human | CHO-K1 | C1038-1a | DC1038-1a | MC1038-1a |
| Cholecystokinin | CCK1 | Human | HEK293T | C1038 | DC1038 | MC1038 |
| Cholecystokinin | CCK2 | Human | HEK293T | H1039 | DH1039 | MH1039 |
| Chemokine | CCR1 | Human | HEK293T | C1009 | DC1009 | MC1009 |
| Chemokine | CCR1 | Human | HEK293T Gαqi5 | CG1009 | DCG1009 | MCG1009 |
| Chemokine | CCR2 | Human | HEK293T | C1010 | DC1010 | MC1010 |
| Chemokine | CCR3 | Human | HEK293T | C1011 | DC1011 | MC1011 |
| Chemokine | CCR3 | Human | HEK293T | CG1011 | DCG1011 | MCG1011 |
| Chemokine | CCR4 | Human | HEK293T | C1012 | DC1012 | MC1012 |
| Chemokine | CCR4 | Human | HEK293T Gαqi5 | CG1012 | DCG1012 | MCG1012 |
| Chemokine | CCR5 | Human | HEK293T | C1013a | DC1013a | MC1013a |
| Chemokine | CCR5 | Human | HEK293T | C1013b | DC1013b | MC1013b |
| Chemokine | CCR5 | Human | HEK293T | CG1013 | DCG1013 | MCG1013 |
| Chemokine | CCR6 | Human | HEK293T | C1014a | DC1014a | MC1014a |
| Chemokine | CCR6 | mouse | HEK293T | Cm1014 | DCm1014 | MCm1014 |
| Chemokine | CCR7 | Human | HEK293T | C1015 | DC1015 | MC1015 |
| Chemokine | CCR7 | Human | HEK293T Gαqi5 | CG1015 | DCG1015 | MCG1015 |
| Chemokine | CCR8 | Human | HEK293T | C1016 | DC1016 | MC1016 |
| Chemokine | CCR8 | Human | HEK293T | C1016a | DC1016a | MC1016a |
| Chemokine | CCR8 | Human | HEK293T Gαqi5 | CG1016 | DCG1016 | MCG1016 |
| Chemokine | CCR9 | dog | HEK293T Gαqi5 | CGd1017 | DCGd1017 | MCGd1017 |
| Chemokine | CCR9 | Human | HEK293T | C1017 | DC1017 | MC1017 |
| Chemokine | CCR9 | Human | HEK293T | C1017a | DC1017a | MC1017a |
| Chemokine | CCR9 | Human | HEK293T Gαqi5 | CG1017 | DCG1017 | MCG1017 |
| Chemokine | CCR9 | Human | HEK293T Gαqi5 | CG1017A | DCG1017A | MCG1017A |
| Chemokine | CCR9 | mouse | HEK293T | Cm1017 | DCm1017 | MCm1017 |
| Chemokine | CCR9 | mouse | HEK293T Gαqi5 | CGm1017 | DCGm1017 | MCGm1017 |
| Chemokine | CCR9 | Rat | HEK293T Gαqi5 | CGr1017 | DCGr1017 | MCGr1017 |
| Chemokine | CCR10 | Human | CHO-K1 Gαqi5 | CG1018 | DCG1018-1 | MCG1018-1 |
| Chemokine | CMKLR1 | Human | HEK293T | C1147 | DC1147 | MC1147 |
| Chemokine | CMKLR1 | Human | HEK293T Gαqi5 | CG1147 | DCG1147 | MCG1147 |
| Chemokine | CX3CR1 | Human | HEK293T | C1008 | DC1008 | MC1008 |
| Chemokine | CX3CR1 | Human | HEK293T Gαqi5 | CG1008 | DCG1008 | MCG1008 |
| Chemokine | CX3CR1 | Human | HEK293T Gαqi5 | CG1008a | DCG1008a | MCG1008a |
| Chemokine | CX3CR1 | Human | HEK293T Gαqi5 | CG1008b | DCG1008b | MCG1008b |
| Chemokine | CXCR1 | Human | HEK293T | C1001a | DC1001a | MC1001a |
| Chemokine | CXCR1 | Human | HEK293T Gαqi5 | CG1001 | DCG1001 | MCG1001 |
| Chemokine | CXCR2 | Human | HEK293T | C1002 | DC1002 | MC1002 |
| Chemokine | CXCR2 | Human | HEK293T Gαqi5 | CG1002 | DCG1002 | MCG1002 |
| Chemokine | CXCR3 | Human | HEK293T | C1003 | DC1003 | MC1003 |
| Chemokine | CXCR3 | Human | HEK293T Gαqi5 | CG1003 | DCG1003 | MCG1003 |
| Chemokine | CXCR4 | Human | HEK293T | C1004-1 | DC1004-1 | MC1004-1 |
| Chemokine | CXCR4 | Human | HEK293T Gαqi5 | CG1004 | DCG1004 | MCG1004 |
| Chemokine | CXCR5 | Human | HEK293T | C1005 | DC1005 | MC1005 |
| Chemokine | CXCR5 | Human | CHO-K1 | C1005-1 | DC1005-1 | MC1005-1 |
| Chemokine | CXCR5 | Human | CHO-K1 | C1005-1a | DC1005-1a | MC1005-1a |
| Chemokine | CXCR6 | Human | HEK293T | C1006 | DC1006 | MC1006 |
| Chemokine | CXCR6 | Human | CHO-K1 | C1006-1 | DC1006-1 | MC1006-1 |
| Chemokine | CXCR6 | Human | HEK293T Gαqi5 | CG1006 | DCG1006 | MCG1006 |
| Chemokine | CXCR7 | Human | HEK293T | C1150 | DC1150 | MC1150 |
| Chemokine | XCR1 | Human | HEK293T | C1007 | DC1007 | MC1007 |
| Cannabinoid | CB1 | Human | HEK293T | C1229 | DC1229 | MC1229 |
| Cannabinoid | CB1 | Human | CHO-K1 | C1229-1a | DC1229-1a | MC1229-1a |
| Cannabinoid | CB1 | Human | CHO-K1 | C1229-1 | DC1229-1 | MC1229-1 |
| Cannabinoid | CB2 | Human | CHO-K1 | C1230-1 | DC1230-1 | MC1230-1 |
| Cannabinoid | CB2 | Human | CHO-K1 | C1230-1a | DC1230-1a | MC1230-1a |
| Cannabinoid | GPR55 | Human | HEK293T | H1113 | DH1113 | MH1113 |
| Cannabinoid | GPR55 | Human | HEK293T | C1113b | DC1113b | MC1113b |
| Calcium-Sensing | CaSR | Human | HEK293T | C1233 | DC1233 | MC1233 |
| Calcium-Sensing | CaSR | Rat | HEK293T | Cr1233 | DCr1233 | MCr1233 |
| Calcitonin | CALCRL | Human | HEK293T | C1232 | DC1232 | MC1232 |
| Calcitonin | CT | Human | HEK293T | H1231 | DH1231 | MH1231 |
| Bradykinin | B1 | Human | HEK293T | C1198a | DC1198a | MC1198a |
| Bradykinin | B1 | mouse | HEK293T | Cm1198 | DCm1198 | MCm1198 |
| Bradykinin | B2 | Human | HEK293T | H1199 | DH1199 | MH1199 |
| Bradykinin | B2 | mouse | HEK293T | Cm1199 | DCm1199 | MCm1199 |
| Bradykinin | B2 | Rat | HEK293T | Cr1199 | DCr1199 | MCr1199 |
| Bradykinin | B2 | dog | HEK293T | Cd1199 | DCd1199 | MCd1199 |
| Bradykinin | B2 | monkey | HEK293T | Cp1199 | DCp1199 | MCp1199 |
| Bradykinin | B2 | guinia pig | HEK293T | Cc1199 | DCc1199 | MCc1199 |
| Bradykinin | B2 | rabbit | HEK293T | Cb1199 | DCb1199 | MCb1199 |
| Bombesin | BB1 | Human | HEK293T | C1211 | DC1211 | MC1211 |
| Bombesin | BB1 | Rat | C6 | C1211-1 | DC1211-1 | MC1211 |
| Bombesin | BB2 | Human | HEK293T | C1215 | DC1215 | MC1211-1 |
| Bombesin | BB3 | Human | HEK293T | C1214 | DC1214 | MC1214 |
| Bombesin | BB3 | Human | HEK293T | H1214 | DH1214 | MH1214 |
| Bile Acid | GPBA | Human | CHO-K1 | C1361-1 | DC1361-1 | MC1361-1 |
| Bile Acid | GPBA | Human | CHO-K1 | C1361-1a | DC1361-1a | MC1361-1a |
| Bile Acid | GPBA | Rat | CHO-K1 | Cr1361-1 | DCr1361-1 | MCr1361-1 |
| Bile Acid | GPBA | mouse | CHO-K1 | Cm1361-1 | DCm1361-1 | MCm1361-1 |
| Apelin | APJ | Human | HEK293T | C1196a | DC1196a | MC1196a |
| Apelin | APJ | Human | CHO-K1 | C1196-1 | DC1196-1 | MC1361-1 |
| Angiotensin | AT1 | Human | HEK293T | H1417 | DH1417 | MH1417 |
| Anaphylatoxin | C3AR1 | Human | HEK293T | C1222 | DC1222 | MC1222 |
| Anaphylatoxin | C5R1 | Human | HEK293T | C1221 | DC1221 | MC1221 |
| Adrenergic | alpha1A | Human | CHO-K1 | C1431-1 | DC1431-1 | MC1431-1 |
| Adrenergic | alpha1B | Human | CHO-K1 | C1432-1 | DC1432-1 | MC1432-1 |
| Adrenergic | alpha1D | Human | CHO-K1 | C1433-1 | DC1433-1 | MC1433-1 |
| Adrenergic | alpha1D | Human | CHO-K1 | C1433-1a | DC1433-1 | MC1433-1a |
| Adrenergic | alpha2A | Human | CHO-K1 | C1434-1 | DC1434-1 | MC1434-1 |
| Adrenergic | alpha2A | Human | CHO-K1 | C1434-1a | DC1434-1a | MC1434-1a |
| Adrenergic | alpha2B | Human | CHO-K1 | C1435-1 | DC1435-1 | MC1435-1 |
| Adrenergic | alpha2C | Human | CHO-K1 | C1436-1 | DC1436-1 | MC1436-1 |
| Adrenergic | beta1 | Human | HEK293T | H1437 | DH1437 | MC1437-1 |
| Adrenergic | beta1 | Human | CHO-K1 | C1437-1 | DC1437-1 | MH1437 |
| Adrenergic | beta2 | Human | CHO-K1 | C1438-1a | DC1438-1a | MC1438-1a |
| Adrenergic | beta3 | Human | HEK293T | C1439a | DC1439a | MC1439a |
| Adhesion Class GPCRs | GPR97 | Human | HEK293R | C1396 | DC1397 | MC1397 |
| Adenosine | A1 | Human | CHO-K1 | C1427-1 | DC1427-1 | MC1427-1 |
| Adenosine | A2A | Human | CHO-K1 | C1428-1 | DC1428-1 | MC1428-1 |
| Adenosine | A2B | Human | HEK293T | C1429 | DC1429 | MC1429 |
| Adenosine | A2B | Rat | HEK293T | Cr1429 | DCr1429 | MCr1429 |
| Adenosine | A3 | Human | HEK293T | C1430 | DC1430 | MC1430 |
